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Hydroxytamoxifen是什么

Web友情链接: 医学导航 医学百科 基因123 中华养生网 本站部分文字及图片均来自于网络,如有侵权及时通知我们,联系邮箱:[email protected] 医学导航 医学百科 基因123 中华 … Web960化工网为您提供4-羟基他莫昔芬 68047-06-3化学品安全技术说明书,4-羟基他莫昔芬msds,包含高清的4-羟基他莫昔芬 68047-06-3结构式图片,包括中文名称、英文名称、别名、分子式、分子量、熔点、密度、蒸汽压、溶解性、外观与性状、用途等说明信息,找化学品安全技术说明书 上960化工网,全国免费 ...

Afimoxifene - Wikipedia

WebTamoxifen, sold under the brand name Nolvadex among others, is a selective estrogen receptor modulator used to prevent breast cancer in women and treat breast cancer in … Web4-Hydroxytamoxifen是tamoxifen的活性代谢产物,是一种选择性的雌激素受体调节分子,在乳腺癌的治疗和化学疗法中应用广泛。 注:本品仅可用于科研实验,严禁用于临床医疗 … creed setzer https://flightattendantkw.com

什么是(4-OHT)有人懂吗?? - 百度知道

WebCAS Number Chemical Formula Molecular Weight Purity Grade 68047-06-3 C 26 H 29 NO 2: 387.51 ≥94% Reagent grade WebChemicalBook 为您提供枸橼酸他莫昔芬(54965-24-1)的化学性质,熔点,沸点,密度,分子式,分子量,物理性质,毒性,结构式,海关编码等信息,同时您还可以浏览枸橼酸他 … WebAlthough it is an antagonist of ER action in breast tissue, it acts as an ER agonist in bone and blood vessels and a partial ER agonist in uterine tissues. α-hydroxy Tamoxifen is a … buck rogers in the 25th century radio

4-Hydroxytamoxifen 4-羟基他莫昔芬 Cas# 68392-35-8 - GlpBio

Category:4-Hydroxytamoxifen Estrogen Receptor/ERR

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Hydroxytamoxifen是什么

Afimoxifene: Uses, Interactions, Mechanism of Action - DrugBank

Webα-Hydroxytamoxifen is a metabolite of tamoxifen, reacts with DNA in the absence of metabolizing enzymes, and causes formation of DNA adducts [1] . Room temperature in … Web化学物质. 盐酸洛哌丁胺,是一种有机物化合物,分子式为C 29 H 34 Cl 2 N 2 O 2 ,分子量为513.51,白色或黄白色粉末, 用作止泻药 ,治疗 腹泻 。. [1] 中文名. 盐酸洛哌丁胺. …

Hydroxytamoxifen是什么

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Web14 jan. 2024 · 4-羟基三苯氧胺(10,100 nM)能够抑制 [3H]雌二醇与人体8 S雌激素受体的结合 [1]。. 4-羟基三苯氧胺激活内含肽连接的无活性Cas9,减少脱靶的CRISPR介导的基 … Web4-Hydroxytamoxifen is a selective estrogen receptor modulator (SERM). 体外活性. 4-Hydroxytamoxifen can inhibit the [3H]estradiol binding to the estrogen receptor (IC50: …

Web14 jan. 2024 · (E)-4-羟基他莫昔芬用途 (E)-4-Hydroxytamoxifen 是 (Z)-4-hydroxytamoxifen 的低活性异构体,是雌激素受体 (estrogen receptor) 调节剂。 产品性质 图谱 (E)-4-羟基他莫昔芬名称 (E)-4-羟基他莫昔芬生物活性 (E)-4-羟基他莫昔芬物理化学性质 (E)-4-羟基他莫昔芬合成线路 (E)-4-羟基他莫昔芬英文别名 4- [1- [4- [2- …

Web31 aug. 2011 · 4-Hydroxytamoxifen 4-羟基他莫昔芬 (Z)-4- (1- [4- (二甲基氨基乙氧基)苯基]-2-苯基-1-丁烯)苯酚 它是雌激素受体拮抗剂 参考资料: baidu 4 评论 分享 举报 Web14 jan. 2024 · 4-羟基他莫西芬文献 179. Combined histone deacetylase inhibition and tamoxifen induces apoptosis in tamoxifen-resistant breast cancer models, by reversing …

WebTamoxifen is a prodrug that is metabolized to active metabolites 4-hydroxytamoxifen (4-OHT) and endoxifen by cytochrome P450 isoforms CYP2D6 and CYP3A4. In breast …

Web(Z)-4-hydroxy Tamoxifen 是一种口服具有活力的雌激素受体选择性调节剂 (SERM)。 它基于 ER 介导的细胞核易位诱导 CRISPR/Cas9 系统。 陶术生物的所有产品和服务仅用于科学研究,我们不为任何个人用途提供产品和服务。 CAS:68047-06-3 加入购物车 大包装询单有特惠! 技术资料 更多批次查询请联系客服 选择批次 纯度:99.37% 生物活性 化学信息 储存和 … creed s haymond ddsWebEndoxifen wordt gezien als de belangrijkste metaboliet, mede omdat de steady-state serumconcentratie van endoxifen ongeveer vijfmaal hoger is dan de concentratie van 4-hydroxytamoxifen. De behandeling met tamoxifen – waarbij nu iedereen in principe 20 mg krijgt – kan mogelijk optimaler door individueel te doseren op basis van de concentraties … creed sheffieldWeb4-Hydroxytamoxifen 4-羟基他莫昔芬 (Z)-4- (1- [4- (二甲基氨基乙氧基)苯基]-2-苯基-1-丁烯)苯酚 它是雌激素受体拮抗剂 解析看不懂? 免费查看同类题视频解析 查看解答 相似问题 … buck rogers in the 25th century s2 e11Web13 jun. 2005 · Afimoxifene (4-Hydroxytamoxifen, trade name TamoGel) is a new estrogen inhibitor under investigation for a variety of estrogen-dependent conditions, including cyclic breast pain and gynecomastia. TamoGel is formulated using Enhanced Hydroalcoholic Gel (EHG) Technology. This technology enables percutaneous delivery of drugs that cannot … creeds firewoodWeb上海南方模式生物科技股份有限公司 www.modelorg.com 400-728-0660 1/3 Tamoxifen诱导Cre-ERT2小鼠 使用指南 Cre-ERT2在无Tamoxifen诱导的情况下,在细胞质内处于无活性 … creed she wears a coat of colors lyricsWeb百度百科是一部内容开放、自由的网络百科全书,旨在创造一个涵盖所有领域知识,服务所有互联网用户的中文知识性百科全书。在这里你可以参与词条编辑,分享贡献你的知识。 buck rogers in the 25th century season 1 castWebHowever, long-term usage of tamoxifen has been linked to increased risk of developing endometrial cancer in women. One of the suggested pathways leading to the potential toxicity of tamoxifen involves its oxidative metabolism to 4-hydroxytamoxifen, which may be further oxidized to an electrophilic quinone methide. buck rogers in the 25th century season 3